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CHIR-99021

  • CAS No:252917-06-9 3-Pyridinecarbonitrile,6-[[2-[[4-(2,4-dichlorophenyl)-5-(5-methyl-1H-imidazol-2-yl)-2-pyrimidinyl]amino]ethyl]amino]-
    Molecular Structure

    Detailed Description

    CHIR-99021CHIR-99021 (CT99021) is a GSK-3α/β inhibitor with IC50 of 10 nM/6.7 nM; > 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.

    IC50 value: 10 nM/6.7 nM for GSK-3α/β [1]

    Target: GSK-3α/β

    in vitro: CHIR-99021 shows greater than 500-fold selectivity for GSK-3 versus its closest homologs CDC2 and ERK2, as well as other protein kinases.

    Target:/products

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