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GSK 525762A

  • Purity: >98%
  • Place of Orign: Princeton,New Jersey,United States
Ms.James Gao

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Item specifics

  • Product Name.:GSK 525762A
  • CAS No: 1260907-17-2

Details

GSK 525762AGSK 525762A (I-BET 762) is an inhibitor for BET proteins with IC50 of ~35 nM.

IC50 Value: ~35 nM

Target: BET

in vitro: GSK 525762A is an inhibitor for BET (bromodomain and extra terminal domain) proteins, BRD2, BRD3 and BRD4, binds to the tandem bromodomains of BET with Kd of 50.5-61.3 nM, displaces a tetra-acetylated H4 peptide prebound to tandem bromodomains of BET with IC50 of 32.5-42.5 nM in FRET analysis.

Target:EGFR

Product Links:http://www.medchemexpress.cn/gsk-525762a.html

Permanent link:http://www.medchemexpress.com/gsk-525762a.html

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