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CAS No 28797-61-7 , Pirenzepine

  • Name: Pirenzepine
  • Synonyms: Gastrozepin;Pirenzepine; 11-[2-(4-Methylpiperazin-1-yl)acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one;
  • CAS Registry Number:
  • Melting Point: 226 - 230 C
  • Flash Point: 281.4°C
  • Boiling Point: 541.7°C at 760 mmHg
  • Flash Point: 281.4°C
  • EINECS: 249-228-4
  • Molecular Weight: 351.41
  • InChI: InChI=1/C19H21N5O2/c1-22-9-11-23(12-10-22)13-17(25)24-16-7-3-2-5-14(16)19(26)21-15-6-4-8-20-18(15)24/h2-8H,9-13H2,1H3,(H,21,26)
  • Molecular Formula: C19H21N5O2
  • Molecular Structure:CAS No:28797-61-7 Pirenzepine

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28797-61-7 Gastrozepin

  • China Shanghai Synnad Chemical Co., Ltd. [Importer/Exporter]
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28797-61-7 Pirenzepine

  • IUPAC NAME-11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one MOLECULAR FORMULA-C19H21N5O2 MOLAR MASS-351.403 g/mol Pirenzepine an M1 selective antagonist, is used in the treatment of peptic ulcers, as it reduce...
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28797-61-7 Pirenzepine

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28797-61-7 Gastrozepin

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28797-61-7 PIRENZEPINE

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References of Pirenzepine
Title: Pirenzepine
CAS Registry Number: 28797-61-7
CAS Name: 5,11-Dihydro-11-[(4-methyl-1-piperazinyl)acetyl]-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Manufacturers' Codes: LS-519
Molecular Formula: C19H21N5O2
Molecular Weight: 351.40
Percent Composition: C 64.94%, H 6.02%, N 19.93%, O 9.11%
Literature References: Tricyclic gastric-acid inhibitor. Prepn: FR 1505795 (1967 to Thomae), C.A. 70, 4154w (1969). Pharmacology: W. Eberlein et al., Arzneim.-Forsch. 27, 356 (1977). Pharmacokinetics: R. Hammes et al., ibid. 928. Mechanism of action: G. Heller et al., Verh. Dtsch. Ges. Inn. Med. 84, 991 (1978), C.A. 90, 132984s (1979). Human pharmacology: H. Brunner et al., Arzneim.-Forsch. 27, 684 (1977). Multicenter controlled clinical trial: Scand. J. Gastroenterol. 17, Suppl. 81, 1-42 (1982). Radioimmunoassay determn in human plasma and urine: C. A. Homon et al., Ther. Drug Monit. 9, 236 (1987). Symposium: ibid. Suppl. 72, 1-273. Review of pharmacology and therapeutic efficacy: A. A. Carmine, R. N. Brogden, Drugs 30, 85-126 (1985). Comprehensive description: H. A. El-Obeid et al., Anal. Profiles Drug Subs. 16, 445-506 (1987).
 
Derivative Type: Dihydrochloride
CAS Registry Number: 29868-97-1
Manufacturers' Codes: LS-519-Cl2
Trademarks: Duogastral (ISM); Durapirenz (Durachemie); Gasteril (Ripari-Gero); Gastrozepin (Thomae); Leblon (De Angeli); Maghen (Savio); Renzepin (Bergamon); Tabe (Bernabo); Ulcuforton (Plantorgan); Ulcosan (Domp?
Molecular Formula: C19H21N5O2.2HCl
Molecular Weight: 424.32
Percent Composition: C 53.78%, H 5.46%, N 16.50%, O 7.54%, Cl 16.71%
Properties: Sol in water, slightly sol in methanol. Practically insol in ether.
 
Therap-Cat: Antiulcerative.
Keywords: Antiulcerative.