Fareston (Toremifene Citrate)
CAS:89778-27-8
Molecular Formula: C26H28ClNO.C6H8O7
Assay: 97.0%~103.0%
Appearance: White crystalline powder.
MF:C26H28ClNO·C6H8O7
MW:598.09
Appearance: White powder
Melting Point: 158-164 oC
Usage:Originally developed to fight breast cancer, bodybuilders have used Fareston to successfully fight gynocomastia caused when testosterone converts to estrogen in the body and men grow breasts.
Description:
Toremifene citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body.
Toremifene citrate is FDA-approved for use in advanced (metastatic) breast cancer. It is also being evaluated for prevention of prostate cancer under the brand name Acapodene.
Toremifene has already been covered that Toremifene is a SERM, and serves to block Estrogen at various receptor sites in certain tissues within the body . As a layman explanation.
Toremifene pretends to be a fake Estrogen that occupies Estrogen receptors within breast tissue. With these receptors occupied by Toremifene, real Estrogen cannot perform their jobs there.
Application:
Toremifene citrate is an oral selective estrogen receptor modulator (SERM) which helps oppose the actions of estrogen in the body. Licensed in the United States under the brand name Fareston, toremifene citrate is FDA-approved for use in advanced (metastatic) breast cancer. It is also being evaluated for prevention of prostate cancer under the brand name Acapodene.
It has already been covered that Toremifene is a SERM, and serves to block Estrogen at various receptor sites in certain tissues within the body (breast tissue in particular). As a layman explanation, Toremifene pretends to be a 'fake' Estrogen that occupies Estrogen receptors within breast tissue. With these receptors occupied by Toremifene, real Estrogen cannot perform their jobs there. Toremifene does not reduce total blood plasma levels of Estrogen. In addition to being antagonistic to Estrogen receptors in breast tissue, it is also antagonistic to Estrogen at the hypothalamus gland (this essentially 'tricks' the hypothalamus into thinking there is little or no circulating Estrogen levels in the body, causing it to increase its manufacture of Testosterone so that it can utilize aromatization to restore these levels.
Toremifene is also agonistic to Estrogen receptors in other tissues in the body (within the liver in particular). This means that whileToremifene will act as an anti-estrogen in breast tissue and the hypothalamus, it will act as an Estrogen within the liver. This can have beneficial impacts especially during an anabolic steroid cycle, such as improving and shifting cholesterol levels into a more favorable range.
Packing:
Discreet packing ways as your requirement, 100% go through.
Storage:
Store in cool and dry area and keep away from direct sunlight.
Advantage:
1. more than 5years Rich experience:Our company is a professional production leading factory in China in pharmaceutical area of many years.
2. Discreet package :The packing suits you best would be choosen to cross customs safely. also our warehouse have more than 1hundreds of packing methods ,Or if you have your own ideal way, it could be also taken into consideration .
3. Top quality. High quality guaranteed, once any problem is found, the package would be reshipped for you .and some other products for free .
4. Security Shipping:Shipping by express (FedEx,UPS,DHL,EMS), by air.The most professional forwarder would be recommanded for you.
5. Fast delivery:we hare stock ,so we can deliver your order in 4hours when payment information was confirmed.
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7. Competitive prices:big discount under market price ,plz connect me ,a gift is ready for you
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