Quick Details:
Formestane
Alias: Formestane; -Hydroxyandrost-4-ene-3,17-dione
CAS NO: 566-48-3
Molecular weight: 302.4126
Molecular formula: C19H26O3
Assay:98%
Purity: 99%
Density:1.19 g/cm3
Melting Point:199-202 °C
Boiling Point:475.4 °C at 760 mmHg
Flash Point:255.4 °C
Storage: Shading, confined preservation
Packing: Foil bag
Chemical Properties: Needles
Usage: An antitumor drug. An aromatase inhibitor .Formestane (Lentaron) is considered a pretty potent steroidal aromatose inhibitor. It is used in the treatment of estrogen-receptor positive breast cancer in post-menopausal women.
Formestane is often used to suppress estrogen production from prohormones. It also acts as a prohormone to 4-hydroxytestosterone, an active steroid which displays weak androgenic activity in addition to acting as a mild aromatase inhibitor.
Application: Transdermally or Orally, take 50-100mg of Formestane per day.
Product Description:
A. Formestane is a synthetic steroidal substance with antineoplastic activity. Formestane binds irreversibly to and inhibits the enzyme aromatase, thereby blocking the conversion of cholesterol to pregnenolone and the peripheral aromatization of androgenic precursors into estrogens.
B. Formestane is a drug that has been previously used in breast cancer treatment. Like most drugs which have some sort of phsyique usage, athletes eventually get a hold of it. Formestane is currently one of the best legal anti-estrogens out there. It is classified as an irreversible arromatase inhibitor, meaning, it destroys the aromatase enzyme.
C. Formestane is often used to suppress estrogen production from anabolic steroids or prohormones. It also acts as a prohormone to 4-hydroxytestosterone, an active steroid which displays weak androgenic activity in addition to acting as a mild aromatase inhibitor.
Background:
Formestane is a drug that has been previously used in breast cancer treatment. Like most drugs which have some sort of phsyique usage, athletes eventually get a hold of it. Formestane is currently one of the best legal anti-estrogens out there. It is classified as an irreversible arromatase inhibitor, meaning, it destroys the aromatase enzyme.
How to Use:
Formestane has a very long active life on the order of 24-36 hours. For most users, a 100mg capsule in the morning, and another at night before bed will work well to keep a good deal of water off you. Again, it depends on your susceptibility to aromatization and what drugs and dosages of anabolics you are using. Never the less, this should suffice for most. Remember, formestane attacks the aromatase enzyme and is therefore a first line inhibitor. So if you need immediate relief of estrogen during your cycle, you need a second class drug (estrogen receptor blocker) such as nolvadex or clomid. Formestane is a lot like arimidex in its mechanism of action in attacking the aromatase enzyme itself.
Superiority
Estrogen is a female sex hormone, produced by the ovaries and placenta. Adrenal cortex also produced a few estrogen. Female children after puberty ovarian secretion of estrogen, start, in order to promote the vagina, uterus, fallopian tube and ovary itself development, at the same time caused menstrual endometrial hyperplasia. Estrogen can promote the subcutaneous fat accumulation, plump; hyperplasia of the breast, nipple, areola dark colors, and produce sexual desire; to promote the body sodium and water retention, bone calcium deposition
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