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CAS No 81982-32-3 , alpiropride

  • Name: alpiropride
  • Synonyms: 5-(Methylaminosulfonyl)-N-[(1-allyl-2-pyrrolidinyl)methyl]-2-methoxy-4-aminobenzamide;alpiropride;RIV 2093;
  • CAS Registry Number:
  • Flash Point: °C
  • Boiling Point: °Cat760mmHg
  • Density: 1.227g/cm3
  • Refractive index: 1.56
  • Flash Point: °C
  • EINECS: 279-867-4
  • Molecular Weight: 382.482
  • InChI: InChI=1/C17H26N4O4S/c1-4-7-21-8-5-6-12(21)11-20-17(22)13-9-16(26(23,24)19-2)14(18)10-15(13)25-3/h4,9-10,12,19H,1,5-8,11,18H2,2-3H3,(H,20,22)
  • Molecular Formula: C17H26N4O4S
  • Molecular Structure:CAS No:81982-32-3 alpiropride

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81982-32-3 Alpiropride

  • Alpiropride, Min 99%
  • China Finechemie Co., Ltd. [Manufacturer]
  • Tel: +86-23-99186710
  • Fax: +86-23-99186729
  • Address: 28th Floor Mordern Building,New-Tech Zone400020 ChongqingCHINA Chongqing,nullChina
Contact Supplier

81982-32-3 ALPIROPRIDE

  • China Nanjing Chemlin Chemical Industry Co.,Ltd. [Manufacturer]
  • Tel: +86 25 8369-7070/ +86 138 51816776 (Mobile)
  • Fax: +86 25 8345-3275
  • Address: Rm.902 Longyin Plaza,
    No. 217 Zhongshan Rd.
    (N)Nanjing 210009,China null,nullChina
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References of alpiropride
Title: Alpiropride
CAS Registry Number: 81982-32-3
CAS Name: 4-Amino-2-methoxy-5-[(methylamino)sulfonyl]-N-[[1-(2-propenyl)-2-pyrrolidinyl]methyl]benzamide
Synonyms: (±)-N-[(1-allyl-2-pyrrolidinyl)methyl]-4-amino-5-(methylsulfamoyl)-o-anisamide; N-(1-allyl-2-pyrrolidinylmethyl)-2-methoxy-4-amino-5-methylsulfamoylbenzamide
Manufacturers' Codes: RIV-2093
Trademarks: Rivistel (Delagrange)
Molecular Formula: C17H26N4O4S
Molecular Weight: 382.48
Percent Composition: C 53.38%, H 6.85%, N 14.65%, O 16.73%, S 8.38%
Literature References: Dopamine D2-receptor antagonist structurally similar to sulpiride, q.v. Prepn: J. Perrot, M. Thominet, EP 47207; eidem, US 4550179 (1982, 1985 both to Soc. d'Etudes Sci. Ind. l'Ile-de-France). Dopamine receptor binding study: P. Sokoloff et al., Arch. Pharmacol. 327, 221 (1984). HPLC determn in plasma and urine: F. Bressolle et al., J. Chromatogr. 343, 443 (1985). Pharmacokinetics and metabolism in humans: F. Bressolle et al., J. Pharm. Clin. 4, 261 (1985). Preliminary study in experimentally induced migraine: A. Bès et al., Int. J. Clin. Pharmacol. Res. 6, 189 (1986).
Properties: Crystals from absolute ethanol, mp 168.5-169°. LD50 in male mice (mg/kg): 44 i.v.; 184 i.p.; 204 s.c.; 3600 orally (Perrot, Thominet, 1985).
Melting point: mp 168.5-169°
Toxicity data: LD50 in male mice (mg/kg): 44 i.v.; 184 i.p.; 204 s.c.; 3600 orally (Perrot, Thominet, 1985)
Therap-Cat: Antimigraine.
Keywords: Antimigraine.